Albuterol and Levalbuterol interaction

Albuterol and Levalbuterol: both prescribing labels flag this combination with the strongest language, such as a contraindication, a boxed warning, or an instruction to avoid it.

Major

Do not combine without a prescriber's guidance. The label language below is the strongest FDA uses.

What the FDA labels say

From the Albuterol (Albuterol Sulate HFA) label · effective 2026-01-30

Major

Other short-acting sympathomimetic aerosol bronchodilators should not be used concomitantly with albuterol.

Drug interactionsby drug classView label on DailyMed
Moderate

Therefore, Albuterol Sulfate HFA, like all other sympathomimetic amines, should be used with caution in patients with underlying cardiovascular disorders, especially coronary insufficiency, cardiac arrhythmias, and hypertension.

Warnings and precautionsby drug classView label on DailyMed
Moderate

Coexisting Conditions Albuterol Sulfate HFA, like other sympathomimetic amines, should be used with caution in patients with convulsive disorders, hyperthyroidism, or diabetes mellitus and in patients who are unusually responsive to sympathomimetic amines.

Warnings and precautionsby drug classView label on DailyMed
Minor

Use of Anti-inflammatory Agents The use of beta-adrenergic agonist bronchodilators alone may not be adequate to control asthma in many patients.

Warnings and precautionsby drug classView label on DailyMed
Minor

Cardiovascular Effects Albuterol Sulfate HFA, like all other beta 2 -adrenergic agonists, can produce clinically significant cardiovascular effects in some patients such as changes in pulse rate or blood pressure.

Warnings and precautionsby drug classView label on DailyMed

From the Levalbuterol (XOPENEX HFA) label · effective 2025-06-02

Major

XOPENEX HFA is contraindicated in patients with a history of hypersensitivity to levalbuterol, racemic albuterol, or any other component of XOPENEX HFA.

Contraindicationsnames AlbuterolView label on DailyMed
Major

Hypersensitivity to levalbuterol, racemic albuterol or any other component of XOPENEX HFA Inhalation Aerosol.

Contraindicationsnames AlbuterolView label on DailyMed
Major

Other short-acting sympathomimetic aerosol bronchodilators or epinephrine should not be used concomitantly with XOPENEX HFA.

Drug interactionsby drug classView label on DailyMed
Moderate

Large doses of intravenous racemic albuterol have been reported to aggravate preexisting diabetes mellitus and ketoacidosis.

Warnings and precautionsnames AlbuterolView label on DailyMed
Moderate

Monoamine oxidase inhibitors (MAOs) or tricyclic antidepressants : May potentiate effect of albuterol on the cardiovascular system.

Drug interactionsnames AlbuterolView label on DailyMed

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Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.