Amiodarone and Orlistat interaction

Amiodarone and Orlistat: the Orlistat prescribing label describes an interaction that usually calls for monitoring, a dose change, or spacing the doses.

Moderate

Usually manageable with monitoring or a dose change. Tell your pharmacist you take both.

What the FDA labels say

From the Orlistat label · effective 2026-01-09

Moderate

Drug Interactions and Decreased Vitamin Absorption ORLISTAT may interact with concomitant drugs including cyclosporine, levothyroxine, warfarin, amiodarone, antiepileptic drugs, and antiretroviral drugs [see Drug Interactions (7) ].

Warnings and precautionsnames AmiodaroneView label on DailyMed
Moderate

Amiodarone: A reduction in exposure to amiodarone was observed when ORLISTAT was co-administered.

Drug interactionsnames AmiodaroneView label on DailyMed
Moderate

Amiodarone A pharmacokinetic study, where amiodarone was orally administered during orlistat treatment, demonstrated a reduction in exposure to amiodarone and its metabolite, desethylamiodarone [see Clinical Pharmocology (12.3) ] .

Drug interactionsnames AmiodaroneView label on DailyMed
Moderate

A reduced therapeutic effect of amiodarone is possible.

Drug interactionsnames AmiodaroneView label on DailyMed
Minor

The effect of commencing orlistat treatment in patients on stable amiodarone therapy has not been studied.

Drug interactionsnames AmiodaroneView label on DailyMed

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Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.