Asenapine and Fluvoxamine interaction

Asenapine and Fluvoxamine: both prescribing labels describe an interaction that usually calls for monitoring, a dose change, or spacing the doses.

Moderate

Usually manageable with monitoring or a dose change. Tell your pharmacist you take both.

What the FDA labels say

From the Asenapine (SAPHRIS) label · effective 2025-01-31

Moderate

Marginal increase of asenapine exposure was observed when SAPHRIS is used with fluvoxamine at 25 mg administered twice daily [ see Clinical Pharmacology ( 12.3 )] .

Drug interactionsnames FluvoxamineView label on DailyMed
Moderate

However, the tested fluvoxamine dose was suboptimal.

Drug interactionsnames FluvoxamineView label on DailyMed
Moderate

Full therapeutic dose of fluvoxamine is expected to cause a greater increase in asenapine exposure.

Drug interactionsnames FluvoxamineView label on DailyMed
Minor

Strong CYP1A2 Inhibitors (e.g., Fluvoxamine) SAPHRIS is metabolized by CYP1A2.

Drug interactionsby drug classView label on DailyMed

From the Fluvoxamine (fluvoxamine maleate) label · effective 2026-04-23

Moderate

CNS Active Drugs Antipsychotics: See Warnings and Precautions ( 5.2 ) .

Drug interactionsby drug classView label on DailyMed

Taking more than these two? Interactions stack. Check your whole list at once; it stays in your browser.

Open in the checker

Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.