Esomeprazole and Tacrolimus interaction

Esomeprazole and Tacrolimus: the Esomeprazole prescribing label describe an interaction that usually calls for monitoring, a dose change, or spacing the doses.

Moderate

Usually manageable with monitoring or a dose change. Tell your pharmacist you take both.

What the FDA labels say

From the Esomeprazole (NEXIUM) label · effective 2025-12-19

Moderate

Tacrolimus Clinical Impact: Potentially increased exposure of tacrolimus, especially in transplant patients who are intermediate or poor metabolizers of CYP2C19.

Drug interactionsnames TacrolimusView label on DailyMed
Moderate

Intervention: Monitor tacrolimus whole blood concentrations and consider reducing the dose, if needed, to maintain therapeutic drug concentrations.

Drug interactionsnames TacrolimusView label on DailyMed
Minor

See prescribing information for tacrolimus.

Drug interactionsnames TacrolimusView label on DailyMed

Taking more than these two? Interactions stack. Check your whole list at once; it stays in your browser.

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Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.