Isosorbide dinitrate and Sildenafil interaction

Isosorbide dinitrate and Sildenafil: both prescribing labels flag this combination with the strongest language, such as a contraindication, a boxed warning, or an instruction to avoid it.

Major

Do not combine without a prescriber's guidance. The label language below is the strongest FDA uses.

What the FDA labels say

From the Isosorbide dinitrate label · effective 2020-03-02

Major

Do not use Isosorbide Dinitrate in patients who are taking certain drugs for erectile dysfunction (phosphodiesterase inhibitors), such as sildenafil, tadalafil, or vardenafil.

Contraindicationsby drug classView label on DailyMed
Major

Concomitant use of Isosorbide Dinitrate with phosphodiesterase inhibitors in any form is contraindicated (see CONTRAINDICATIONS ).

Drug interactionsby drug classView label on DailyMed
Moderate

WARNINGS Amplification of the vasodilatory effects of Isosorbide Dinitrate by sildenafil can result in severe hypotension.

Warningsnames SildenafilView label on DailyMed

From the Sildenafil label · effective 2026-07-17

Major

CONTRAINDICATIONS Administration of SILDENAFIL ORAL FILM to patients using nitric oxide donors, such as organic nitrates or organic nitrites in any form.

Contraindicationsby drug classView label on DailyMed
Major

SILDENAFIL ORAL FILM was shown to potentiate the hypotensive effect of nitrates.

Contraindicationsby drug classView label on DailyMed
Major

…its known effects on the nitric oxide/cGMP pathway [see Clinical Pharmacology ( 12.1 , 12.2 ) ] , SILDENAFIL ORAL FILM potentiates the hypotensive effects of nitrates, and its administration to patients who are using nitric oxide donors such as organic nitrates or organic nitrites in any form either regularly and/or intermittently is therefore contraindicated.

Contraindicationsby drug classView label on DailyMed
Major

After patients have taken SILDENAFIL ORAL FILM it is unknown when nitrates, if necessary, can be safely administered.

Contraindicationsby drug classView label on DailyMed
Major

Although plasma levels of sildenafil at 24 hours post dose are much lower than at peak concentration, it is unknown whether nitrates can be safely co-administered at this time point [see Dosage and Administration ( 2.2 ), Drug Interactions ( 7.1 ), and Clinical Pharmacology ( 12.2 ) ].

Contraindicationsby drug classView label on DailyMed

Taking more than these two? Interactions stack. Check your whole list at once; it stays in your browser.

Open in the checker

Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.