Zileuton: interakcje

Zileuton (Zyflo), inhibitor CYP1A2: 130 udokumentowanych interakcji w indeksowanych przez nas etykietach FDA i kartach informacyjnych. Poważne: 9, umiarkowane: 45, niewielkie: 54, pary, dla których etykieta nie zgłasza istotnej interakcji: 22. Każda pozycja poniżej cytuje zdanie, na którym się opiera. Ta strona leku to punkt wyjścia, a nie rozstrzygnięcie dla indywidualnej sytuacji.

Interakcje z etykiety

Poważne interakcje (9)

  • AlosetronPoważna

    Fluvoxamine, a known strong inhibitor of CYP1A2, has been shown to increase mean alosetron plasma concentrations (AUC) approximately 6-fold and prolong the half-life by approximately 3-fold [see Drug Interactions ( 7.1 )] . (etykieta leku Alosetron, Przeciwwskazania)

  • DuloksetynaSNRIPoważna

    Strong CYP1A2 inhibitors : Avoid concomitant use. (etykieta leku Duloksetyna, Interakcje z innymi lekami)

  • ErlotynibPoważna

    Reduce the erlotinib dosage when co-administering with a strong CYP3A4 inhibitor or a combined CYP3A4 and CYP1A2 inhibitor if co-administration is unavoidable [see Dosage and Administration (2.4) ]. (etykieta leku Erlotynib, Interakcje z innymi lekami)

  • Pimozydlek przeciwpsychotycznyPoważna

    Other drugs that are relatively less potent inhibitors of CYP 3A4 should also be avoided, in view of the risks: e.g., zileuton, fluvoxamine. (etykieta leku Pimozyd, Przeciwwskazania)

  • PirfenidonPoważna

    Use of fluvoxamine or other strong CYP1A2 inhibitors should be discontinued prior to administration of ESBRIET and avoided during ESBRIET treatment. (etykieta leku Pirfenidon, Interakcje z innymi lekami)

  • PomalidomidPoważna

    Strong CYP1A2 Inhibitors: Avoid concomitant use of strong CYP1A2 inhibitors. (etykieta leku Pomalidomid, Interakcje z innymi lekami)

  • Ramelteonlek uspokajająco-nasennyPoważna

    Fluvoxamine (strong CYP1A2 inhibitor): Increases AUC for ramelteon and should not be used in combination. (etykieta leku Ramelteon, Przeciwwskazania)

  • Tasimelteonlek uspokajająco-nasennyPoważna

    Strong CYP1A2 inhibitors (e.g., fluvoxamine): Avoid use of HETLIOZ in combination with strong CYP1A2 inhibitors because of increased exposure ( 7.1 , 12.3 ) (etykieta leku Tasimelteon, Interakcje z innymi lekami)

  • Tyzanidynalek zwiotczający mięśniePoważna

    Zanaflex is contraindicated in patients taking strong CYP1A2 inhibitors [see Drug Interactions ( 7.1 )] . with a history of hypersensitivity to tizanidine or the ingredients in Zanaflex. (etykieta leku Tyzanidyna, Przeciwwskazania)

Umiarkowane interakcje (45)

  • Acebutololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • AlkoholAlkoholUmiarkowana

    Use Zileuton Extended-Release Tablets with caution in patients who consume substantial quantities of alcohol and/or have a history of liver disease. (etykieta leku Zileuton, Ostrzeżenia i środki ostrożności)

  • Allopurynolinhibitor oksydazy ksantynowejUmiarkowana

    Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • AminofilinametyloksantynaUmiarkowana

    Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Anagrelidlek wydłużający odstęp QTUmiarkowana

    Drugs that inhibit CYP1A2 (e.g., fluvoxamine, ciprofloxacin) could increase the exposure of AGRYLIN. (etykieta leku Anagrelid, Interakcje z innymi lekami)

  • Atenololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Atenolol + chlortalidonbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • BendamustynaUmiarkowana

    Effect of Other Drugs on Bendamustine Hydrochloride Injection CYP1A2 Inhibitors The coadministration of Bendamustine Hydrochloride Injection with CYP1A2 inhibitors may increase bendamustine plasma concentrations and may result in increased incidence of adverse reactions with Bendamustine Hydrochloride Injection [see Clinical Pharmacology (12.3) ] . (etykieta leku Bendamustyna, Interakcje z innymi lekami)

  • Betaksololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Bisoprololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Bisoprolol + hydrochlorotiazydbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Brymonidyna + tymololagonista receptorów alfa-adrenergicznychUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Dorzolamid + tymololinhibitor anhydrazy węglanowejUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Ergotamina + kofeinaalkaloid sporyszuUmiarkowana

    Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Esmololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Famotydynaantagonista receptora H2Umiarkowana

    Tizanidine (CYP1A2 Substrate) Although not studied clinically, famotidine is considered a weak CYP1A2 inhibitor and may lead to substantial increases in blood concentrations of tizanidine, a CYP1A2 substrate. (etykieta leku Famotydyna, Interakcje z innymi lekami)

  • Febuksostatinhibitor oksydazy ksantynowejUmiarkowana

    Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Ibuprofen + famotydynaNLPZUmiarkowana

    Tizanidine (CYP1A2 Substrate) Clinical Impact Famotidine is considered a weak CYP1A2 inhibitor and may lead to substantial increases in blood concentrations of tizanidine, a CYP1A2 substrate. (etykieta leku Ibuprofen + famotydyna, Interakcje z innymi lekami)

  • Karwedilolbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Klozapinalek przeciwpsychotycznyUmiarkowana

    • Concomitant use of Strong CYP1A2 Inhibitors: Reduce CLOZARIL dose to one-third when coadministered with strong CYP1A2 inhibitors (e.g., fluvoxamine, ciprofloxacin, enoxacin). (etykieta leku Klozapina, Interakcje z innymi lekami)

  • Labetalolbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • LomitapidUmiarkowana

    …Weak CYP3A4 inhibitors (such as alprazolam, amiodarone, amlodipine, atorvastatin, bicalutamide, cilostazol, cimetidine, cyclosporine, fluoxetine, fluvoxamine, ginkgo, goldenseal, isoniazid, lapatinib, nilotinib, pazopanib, ranitidine, ranolazine, ticagrelor, zileuton) can increase lomitapide exposure approximately 2-fold [see Clinical Pharmacology (12.3) ] . (etykieta leku Lomitapid, Interakcje z innymi lekami)

  • Metoprololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Metoprolol + hydrochlorotiazydbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Nadololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Nebiwololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Olanzapinalek przeciwpsychotycznyUmiarkowana

    Inhibitors of CYP1A2 Fluvoxamine: Fluvoxamine, a CYP1A2 inhibitor, decreases the clearance of olanzapine. (etykieta leku Olanzapina, Interakcje z innymi lekami)

  • Olanzapina + fluoksetynalek przeciwpsychotycznyUmiarkowana

    Inhibitors of CYP1A2 — Fluvoxamine decreases the clearance of olanzapine. (etykieta leku Olanzapina + fluoksetyna, Interakcje z innymi lekami)

  • Orfenadryna + kwas acetylosalicylowy + kofeinalek zwiotczający mięśnieUmiarkowana

    Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • PentoksyfilinametyloksantynaUmiarkowana

    Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Pindololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Propranololbeta-blokerUmiarkowana

    Propranolol Co-administration of zileuton immediate-release tablets and propranolol results in a significant increase in propranolol concentrations. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Prymachinalek przeciwmalarycznyUmiarkowana

    Effects of Primaquine on the Pharmacokinetics of Other Drugs CYP1A2 Substrates Published clinical and non-clinical reports indicate primaquine inhibits CYP1A2 enzyme activity and thus may lead to increased exposure of CYP1A2 substrate drugs (e.g., duloxetine, alosetron, theophylline and tizanidine) when co-administered with Primaquine phosphate Tablets. (etykieta leku Prymachina, Interakcje z innymi lekami)

  • Rasagilinainhibitor MAOUmiarkowana

    Ciprofloxacin or Other CYP1A2 Inhibitors Rasagiline plasma concentrations may increase up to 2 fold in patients using concomitant ciprofloxacin and other CYP1A2 inhibitors. (etykieta leku Rasagilina, Ostrzeżenia i środki ostrożności)

  • Ropinirolagonista dopaminyUmiarkowana

    Therefore, if therapy with a drug known to be a potent inducer or inhibitor of CYP1A2 is stopped or started during treatment with ropinirole, adjustment of the dose of ropinirole may be required. (etykieta leku Ropinirol, Interakcje z innymi lekami)

  • Ropiwakainaśrodek znieczulający miejscowoUmiarkowana

    In vivo, the plasma clearance of ropivacaine was reduced by 70% during coadministration of fluvoxamine (25 mg bid for 2 days), a selective and potent CYP1A2 inhibitor. (etykieta leku Ropiwakaina, Interakcje z innymi lekami)

  • RyluzolUmiarkowana

    Strong to moderate CYP1A2 inhibitors: Co-administration may increase TIGLUTIK-associated adverse reactions ( 7.1 ) (etykieta leku Ryluzol, Interakcje z innymi lekami)

  • Sotalolbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • TeofilinametyloksantynaUmiarkowana

    Zileuton increases theophylline levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Tymololbeta-blokerUmiarkowana

    Zileuton increases propranolol levels and beta-blocker activity. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Warfarynalek przeciwzakrzepowyUmiarkowana

    Zileuton increases warfarin levels. (etykieta leku Zileuton, Interakcje z innymi lekami)

Wzmianki o niewielkim znaczeniu (54)

  • Amiodaronlek przeciwarytmicznyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Aprepitantinhibitor CYP3A4Niewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Asenapinalek przeciwpsychotycznyNiewielka

    Strong CYP1A2 Inhibitors (e.g., Fluvoxamine) SAPHRIS is metabolized by CYP1A2. (etykieta leku Asenapina, Interakcje z innymi lekami)

  • Atazanawirlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • BudezonidkortykosteroidNiewielka

    An open-label, nonrandomized clinical study examined the immune responsiveness to varicella vaccine in 243 asthma patients 12 months to 8 years of age who were treated with budesonide inhalation suspension 0.25 mg to 1 mg daily (n=151) or non-corticosteroid asthma therapy (n=92) (i.e., beta 2 -agonists, leukotriene receptor antagonists, cromones). (etykieta leku Budezonid, Ostrzeżenia i środki ostrożności)

  • Budezonid + formoterolkortykosteroidNiewielka

    An open-label, nonrandomized clinical study examined the immune responsiveness to varicella vaccine in 243 asthma patients 12 months to 8 years of age who were treated with budesonide inhalation suspension 0.25 mg to 1 mg daily (n=151) or noncorticosteroid asthma therapy (n=92) (i.e., beta 2 -agonists, leukotriene receptor antagonists, cromones). (etykieta leku Budezonid + formoterol, Ostrzeżenia i środki ostrożności)

  • Cenobamatlek przeciwdrgawkowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Cyklosporynalek immunosupresyjnyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Cymetydynaantagonista receptora H2Niewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Darunawirlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Darunawir + kobicystatlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Digoksynaglikozyd naparstnicyNiewielka

    Drug-drug interaction studies in healthy subjects have been conducted with zileuton immediate-release tablets and digoxin, phenytoin, sulfasalazine, and naproxen. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Dihydroergotaminaalkaloid sporyszuNiewielka

    Less potent inhibitors include saquinavir, nefazodone, fluconazole, grapefruit juice, fluoxetine, fluvoxamine, zileuton, and clotrimazole. (etykieta leku Dihydroergotamina, Ostrzeżenia)

  • Diltiazembloker kanału wapniowegoNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Dronedaronlek przeciwarytmicznyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Efawirenzlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Efawirenz + lamiwudyna + tenofowirlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • ErybulinaNiewielka

    Effect s of HALAVEN on Other Drugs Eribulin does not inhibit CYP1A2, CYP2C9, CYP2C19, CYP2D6, CYP2E1 or CYP3A4 enzymes or induce CYP1A2, CYP2C9, CYP2C19 or CYP3A4 enzymes at relevant clinical concentrations. (etykieta leku Erybulina, Interakcje z innymi lekami)

  • Erytromycynaantybiotyk makrolidowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Ewerolimuslek immunosupresyjnyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Fenytoinalek przeciwdrgawkowyNiewielka

    Drug-drug interaction studies in healthy subjects have been conducted with zileuton immediate-release tablets and digoxin, phenytoin, sulfasalazine, and naproxen. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Flukonazolazolowy lek przeciwgrzybiczyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Fosamprenawirlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Fosaprepitantinhibitor CYP3A4Niewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • GemfibrozylfibratNiewielka

    (E) In vitro studies of CYP enzymes, UGTA enzymes and OATP1B1 transporter In vitro studies have shown that gemfibrozil is an inhibitor of CYP1A2, CYP2C8, CYP2C9, CYP2C19, OATP1B1, and UDP-glucuronosyltransferase (UGT) 1A1 and 1A3 (see WARNINGS ). (etykieta leku Gemfibrozyl, Interakcje z innymi lekami)

  • Imatynibinhibitor CYP3A4Niewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Itrakonazolazolowy lek przeciwgrzybiczyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Iwakaftorinhibitor CYP3A4Niewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • IzoniazydantybiotykNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Karbamazepinalek przeciwdrgawkowyNiewielka

    …voriconazole ) , cimetidine, ciprofloxacin, clarithromycin, dalfopristin, danazol, dantrolene, delavirdine, diltiazem, erythromycin, fluoxetine, fluvoxamine, grapefruit juice, ibuprofen, isoniazid, loratadine, nefazodone, niacinamide, nicotinamide, olanzapine, omeprazole, oxybutynin, quinine, quinupristin, ticlopidine, troleandomycin, valproate, verapamil, zileuton. (etykieta leku Karbamazepina, Interakcje z innymi lekami)

  • Ketokonazolazolowy lek przeciwgrzybiczyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Klarytromycynaantybiotyk makrolidowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Lenakapawirlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Lopinawir + rytonawirlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Mifeprystoninhibitor CYP3A4Niewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Mirabegronagonista receptorów beta-adrenergicznychNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • NaproksenNLPZNiewielka

    Drug-drug interaction studies in healthy subjects have been conducted with zileuton immediate-release tablets and digoxin, phenytoin, sulfasalazine, and naproxen. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Drug-drug interaction studies in healthy subjects have been conducted with zileuton immediate-release tablets and digoxin, phenytoin, sulfasalazine, and naproxen. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Nefazodonlek przeciwdepresyjnyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Nirmatrelwir + rytonawirlek przeciwwirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Palbocyklibinhibitor CYP3A4Niewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Perampanellek przeciwdrgawkowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Pozakonazolazolowy lek przeciwgrzybiczyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Ranolazynalek wydłużający odstęp QTNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Rytlecytynibinhibitor JAKNiewielka

    CYP1A2 Substrates Where Small Concentration Changes May Lead to Serious Adverse Reactions Clinical Impact Ritlecitinib is a CYP1A2 inhibitor. (etykieta leku Rytlecytynib, Interakcje z innymi lekami)

  • Rytonawirlek przeciwretrowirusowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • SulfasalazynasulfonamidNiewielka

    Drug-drug interaction studies in healthy subjects have been conducted with zileuton immediate-release tablets and digoxin, phenytoin, sulfasalazine, and naproxen. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Sumatryptan + naproksentryptanNiewielka

    Drug-drug interaction studies in healthy subjects have been conducted with zileuton immediate-release tablets and digoxin, phenytoin, sulfasalazine, and naproxen. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Suworeksantlek uspokajająco-nasennyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Tikagrelorlek przeciwpłytkowyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • WenlafaksynaSNRINiewielka

    CYP1A2 Venlafaxine did not inhibit CYP1A2 in vitro . (etykieta leku Wenlafaksyna, Interakcje z innymi lekami)

  • Werapamilbloker kanału wapniowegoNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Worykonazolazolowy lek przeciwgrzybiczyNiewielka

    However, no formal drug-drug interaction studies between zileuton and CYP3A4 inhibitors, such as ketaconazole, have been conducted. (etykieta leku Zileuton, Interakcje z innymi lekami)

Nie zgłoszono istotnej interakcji (22)

  • Dezogestrel + etynyloestradioldoustny środek antykoncepcyjnyBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Dioctan etynodiolu + etynyloestradioldoustny środek antykoncepcyjnyBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Drospirenon + etynyloestradioldoustny środek antykoncepcyjnyBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • EstradiolestrogenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Estradiol + dienogestdoustny środek antykoncepcyjnyBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Estradiol + noretysteronestrogenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Estrogeny skoniugowaneestrogenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Etonogestrel + etynyloestradiolestrogenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • FulwestrantestrogenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • LewonorgestrelprogestagenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Lewonorgestrel + etynyloestradioldoustny środek antykoncepcyjnyBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • MedroksyprogesteronprogestagenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • MegestrolprogestagenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Norelgestromin + etynyloestradiolestrogenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • NoretysteronprogestagenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Noretysteron + etynyloestradioldoustny środek antykoncepcyjnyBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Norgestrel + etynyloestradioldoustny środek antykoncepcyjnyBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • Norgestymat + etynyloestradioldoustny środek antykoncepcyjnyBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • PrednizonkortykosteroidBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

  • ProgesteronprogestagenBrak interakcji

    Other Concomitant Drug Therapy Drug-drug interaction studies conducted in healthy subjects between zileuton immediate-release tablets and prednisone and ethinyl estradiol (oral contraceptive), drugs known to be metabolized by the CYP3A4 isoenzyme, have shown no significant interaction. (etykieta leku Zileuton, Interakcje z innymi lekami)

Sprawdź, jak Zileuton łączy się ze wszystkim, co przyjmujesz. Dodaj całą listę; wszystkie pary są sprawdzane jednocześnie.

Otwórz w wyszukiwarce

To nie jest porada medyczna. Stopień nasilenia odzwierciedla sformułowania etykiety, a nie indywidualne okoliczności. Oznaczenie „poważna” może dotyczyć połączenia stosowanego rutynowo pod nadzorem, a „niewielka” może mieć znaczenie przy dużych dawkach. Należy zapytać farmaceutę.