Acetazolamide and Phenytoin interaction

Acetazolamide and Phenytoin: both prescribing labels describe an interaction that usually calls for monitoring, a dose change, or spacing the doses.

Moderate

Usually manageable with monitoring or a dose change. Tell your pharmacist you take both.

What the FDA labels say

From the Acetazolamide label · effective 2026-01-23

Moderate

Acetazolamide modifies phenytoin metabolism with increased serum levels of phenytoin.

Drug interactionsnames PhenytoinView label on DailyMed
Moderate

This may increase or enhance the occurrence of osteomalacia in some patients receiving chronic phenytoin therapy.

Drug interactionsnames PhenytoinView label on DailyMed
Moderate

By decreasing the gastrointestinal absorption of primidone, acetazolamide may decrease serum concentrations of primidone and its metabolites, with a consequent possible decrease in anticonvulsant effect.

Drug interactionsby drug classView label on DailyMed

From the Phenytoin label · effective 2024-12-24

Moderate

…voriconazole Antineoplastic agents Capecitabine, fluorouracil Antidepressants Fluoxetine, fluvoxamine, sertraline Gastric acid reducing agents H 2 antagonists (cimetidine), omeprazole Sulfonamides Sulfamethizole, sulfaphenazole, sulfadiazine, sulfamethoxazole-trimethoprim Other Acute alcohol intake, amiodarone, chloramphenicol, chlordiazepoxide, disulfiram, estrogen,…

Drug interactionsby drug classView label on DailyMed

Taking more than these two? Interactions stack. Check your whole list at once; it stays in your browser.

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Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.