Asenapine and Clonidine interaction

Asenapine and Clonidine: both prescribing labels flag this combination with the strongest language, such as a contraindication, a boxed warning, or an instruction to avoid it.

Major

Do not combine without a prescriber's guidance. The label language below is the strongest FDA uses.

What the FDA labels say

From the Clonidine (QLONILIK) label · effective 2026-08-12

Major

Avoid use with other central nervous system (CNS) depressants ( 5.3 )

Warnings and precautionsby drug classView label on DailyMed
Major

Avoid use with other central nervous system (CNS) depressants, as this combination may cause excessive drowsiness or sedation [see Drug Interactions (7) ].

Warnings and precautionsby drug classView label on DailyMed
Major

Intervention Avoid concomitant use of CNS depressants with QLONILIK.

Drug interactionsby drug classView label on DailyMed
Moderate

Intervention Monitor blood pressure and heart rate, and adjust dosage of QLONILIK accordingly in patients treated concomitantly with antihypertensives CNS depressants Clinical Implication Concomitant use of CNS depressants with clonidine potentiates the sedating effects [see Warnings and Precautions (5.3) ].

Drug interactionsby drug classView label on DailyMed
Moderate

Concomitant use of CNS depressants with clonidine potentiates the sedating effects.

Drug interactionsby drug classView label on DailyMed

From the Asenapine (SAPHRIS) label · effective 2025-01-31

Moderate

Orthostatic vital signs should be monitored in patients who are vulnerable to hypotension (elderly patients, patients with dehydration, hypovolemia, concomitant treatment with antihypertensive medications, patients with known cardiovascular disease (history of myocardial infarction or ischemic heart disease, heart failure, or conduction abnormalities), and patients…

Warnings and precautionsby drug classView label on DailyMed
Moderate

Antihypertensive Drugs: SAPHRIS may cause hypotension.

Drug interactionsby drug classView label on DailyMed
Moderate

…SAPHRIS Table 12: Clinically Important Drug Interactions with SAPHRIS Concomitant Drug Name or Drug Class Clinical Rationale Clinical Recommendation Antihypertensive Drugs Because of its α 1 -adrenergic antagonism with potential for inducing hypotension, SAPHRIS may enhance the effects of certain antihypertensive agents [see Warnings and Precautions ( 5.7 )] .

Drug interactionsby drug classView label on DailyMed
Moderate

Monitor blood pressure and adjust dosage of antihypertensive drug accordingly.

Drug interactionsby drug classView label on DailyMed

Taking more than these two? Interactions stack. Check your whole list at once; it stays in your browser.

Open in the checker

Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.