Fluconazole and Glipizide interaction

Fluconazole and Glipizide: both prescribing labels flag this combination with the strongest language, such as a contraindication, a boxed warning, or an instruction to avoid it.

Major

Do not combine without a prescriber's guidance. The label language below is the strongest FDA uses.

What the FDA labels say

From the Fluconazole label · effective 2026-04-02

Major

Oral hypoglycemics Clinically significant hypoglycemia may be precipitated by the use of fluconazole with oral hypoglycemic agents; one fatality has been reported from hypoglycemia in association with combined fluconazole and glyburide use.

Drug interactionsby drug classView label on DailyMed
Moderate

Fluconazole reduces the metabolism of tolbutamide, glyburide, and glipizide and increases the plasma concentration of these agents.

Drug interactionsnames GlipizideView label on DailyMed
Moderate

When fluconazole is used concomitantly with these or other sulfonylurea oral hypoglycemic agents, blood glucose concentrations should be carefully monitored and the dose of the sulfonylurea should be adjusted as necessary.

Drug interactionsby drug classView label on DailyMed

From the Glipizide (Glucotrol XL) label · effective 2026-07-21

Moderate

Severe hypoglycemia can occur when GLUCOTROL and oral miconazole are used concomitantly ( 7.2 , 12.3 ). ▪ Fluconazole: Monitor patients closely.

Drug interactionsnames FluconazoleView label on DailyMed
Moderate

An increase in GLUCOTROL AUC was seen after fluconazole administration ( 7.3 , 12.3 ). ▪ Colesevelam: GLUCOTROL XL should be administered at least 4 hours prior to colesevelam ( 7.4 , 12.3 ).

Drug interactionsnames FluconazoleView label on DailyMed
Moderate

Fluconazole Monitor patients closely for hypoglycemia when Glucotrol XL is co-administered with fluconazole.

Drug interactionsnames FluconazoleView label on DailyMed
Moderate

Concomitant treatment with fluconazole increases plasma concentrations of glipizide, which may lead to hypoglycemia [see Clinical Pharmacology (12.3) ] .

Drug interactionsnames FluconazoleView label on DailyMed

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Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.