Isosorbide mononitrate and Riociguat interaction

Isosorbide mononitrate and Riociguat: both prescribing labels flag this combination with the strongest language, such as a contraindication, a boxed warning, or an instruction to avoid it.

Major

Do not combine without a prescriber's guidance. The label language below is the strongest FDA uses.

What the FDA labels say

From the Isosorbide mononitrate label · effective 2019-11-01

Major

Do not use isosorbide mononitrate in patients who are taking the soluble guanylate cyclase stimulator riociguat.

Contraindicationsnames RiociguatView label on DailyMed
Major

Concomitant use of isosorbide mononitrate with riociguat, a soluble guanylate cyclase stimulator, is contraindicated (see CONTRAINDICATIONS).

Drug interactionsnames RiociguatView label on DailyMed
Moderate

The vasodilating effects of isosorbide mononitrate may be additive with those of other vasodilators.

Drug interactionsby drug classView label on DailyMed

From the Riociguat (Adempas) label · effective 2026-08-13

Major

• Use with nitrates or nitric oxide donors in any form ( 4.2 , 7.1 )

Contraindicationsby drug classView label on DailyMed
Major

Nitrates and Nitric Oxide Donors Co-administration of Adempas with nitrates or nitric oxide donors (such as amyl nitrite) in any form is contraindicated [see Drug Interactions (7.1) and Clinical Pharmacology (12.2) ] .

Contraindicationsby drug classView label on DailyMed
Major

Nitrates: Co-administration of Adempas with nitrates or nitric oxide donors (such as amyl nitrite) in any form is contraindicated because of hypotension [see Contraindications (4.2) and Clinical Pharmacology (12.2) ] .

Drug interactionsby drug classView label on DailyMed

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Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.