Nitroglycerin and Riociguat interaction

Nitroglycerin and Riociguat: both prescribing labels flag this combination with the strongest language, such as a contraindication, a boxed warning, or an instruction to avoid it.

Major

Do not combine without a prescriber's guidance. The label language below is the strongest FDA uses.

What the FDA labels say

From the Nitroglycerin (NITROGLYCERIN LINGUAL) label · effective 2025-12-17

Major

Use of phosphodiesterase type 5 (PDE-5) Inhibitors, such as avanafil, sildenafil, tadalafil, or vardenafil, or soluble guanylate cyclase (sGC) stimulator (riociguat).

Contraindicationsnames RiociguatView label on DailyMed
Major

Do not use Nitroglycerin Lingual Spray in patients who are taking soluble guanylate cyclase (sGC) stimulators, such as riociguat.

Contraindicationsnames RiociguatView label on DailyMed

From the Riociguat (Adempas) label · effective 2026-08-13

Major

• Use with nitrates or nitric oxide donors in any form ( 4.2 , 7.1 )

Contraindicationsby drug classView label on DailyMed
Major

Nitrates and Nitric Oxide Donors Co-administration of Adempas with nitrates or nitric oxide donors (such as amyl nitrite) in any form is contraindicated [see Drug Interactions (7.1) and Clinical Pharmacology (12.2) ] .

Contraindicationsby drug classView label on DailyMed
Major

Nitrates: Co-administration of Adempas with nitrates or nitric oxide donors (such as amyl nitrite) in any form is contraindicated because of hypotension [see Contraindications (4.2) and Clinical Pharmacology (12.2) ] .

Drug interactionsby drug classView label on DailyMed

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Not medical advice. Interaction Checker quotes FDA label text and NIH fact sheets. Whether an interaction matters for you depends on doses, timing, kidney and liver function, and other conditions. Confirm with a pharmacist or prescriber.