Interações de Tafenoquina

Tafenoquina (Krintafel, Arakoda), antimalárico, tem 34 interações documentadas nas bulas da FDA e nas fichas informativas que indexamos (graves: 12; moderadas: 19; leves: 3; casos em que uma bula relata não haver interação significativa: 0). Cada item abaixo cita a frase em que se baseia. Esta página de medicamento é um ponto de partida, não um veredito para a sua situação.

Interações segundo a bula

Interações graves (12)

  • Alogliptina + metforminainibidor da DPP-4Grave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • Dapagliflozina + metforminainibidor do SGLT2Grave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • DofetilidaantiarrítmicoGrave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • Empagliflozina + metforminainibidor do SGLT2Grave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • Glibenclamida + metforminasulfonilureiaGrave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • Glipizida + metforminasulfonilureiaGrave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • Linagliptina + metforminainibidor da DPP-4Grave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • MetforminabiguanidaGrave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • Penicillamine should not be used in patients who are receiving concurrently gold therapy, antimalarial or cytotoxic drugs, oxyphenbutazone or phenylbutazone because these drugs are also associated with similar serious hematologic and renal adverse reactions. (bula de Penicilamina, Precauções)

  • Pioglitazona + metforminatiazolidinedionaGrave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • Saxagliptina + metforminainibidor da DPP-4Grave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

  • Sitagliptina + metforminainibidor da DPP-4Grave

    Avoid coadministration of ARAKODA with OCT2 and MATE substrates (e.g., dofetilide, metformin). (bula de Tafenoquina, Interações medicamentosas)

Interações moderadas (19)

  • Articaína + epinefrinaanestésico localModerada

    …ropivacaine, tetracaine Antineoplastic agents cyclophosphamide, flutamide, hydroxyurea, ifosfamide, rasburicase Antibiotics dapsone, nitrofurantoin, para-aminosalicylic acid, sulfonamides Antimalarials chloroquine, primaquine Anticonvulsants phenobarbital, phenytoin, sodium valproate Other drugs acetaminophen, metoclopramide, quinine, sulfasalazine Monoamine Oxidase… (bula de Articaína + epinefrina, Interações medicamentosas)

  • Bupivacaínaanestésico localModerada

    • Drugs Associated with Methemoglobinemia : Patients are at increased risk of developing methemoglobinemia when concurrently exposed to nitrates, nitrites, local anesthetics, antineoplastic agents, antibiotics, antimalarials, anticonvulsants, and other drugs. (bula de Bupivacaína, Interações medicamentosas)

  • Bupivacaína + epinefrinaanestésico localModerada

    • Drugs Associated with Methemoglobinemia : Patients are at increased risk of developing methemoglobinemia when concurrently exposed to nitrates, nitrites, local anesthetics, antineoplastic agents, antibiotics, antimalarials, anticonvulsants, and other drugs. (bula de Bupivacaína + epinefrina, Interações medicamentosas)

  • Cloroprocaínaanestésico localModerada

    …procaine, ropivacaine, tetracaine Antineoplastic agents cyclophosphamide, flutamide, hydroxyurea, ifosfamide, rasburicase Antibiotics dapsone, nitrofurantoin, para-aminosalicylic acid, sulfonamides Antimalarials chloroquine, primaquine Anticonvulsants Phenobarbital, phenytoin, sodium valproate Other drugs acetaminophen, metoclopramide, quinine, sulfasalazine (bula de Cloroprocaína, Precauções)

  • CloroquinaantimaláricoModerada

    Patients infected with a resistant strain of plasmodia as shown by the fact that normally adequate doses have failed to prevent or cure clinical malaria or parasitemia should be treated with another form of antimalarial therapy. (bula de Cloroquina, Advertências)

  • DarunavirantirretroviralModerada

    Antimalarial : artemether/lumefantrine ↓ artemether ↓ dihydroartemisinin ↑ lumefantrine ↔ darunavir The combination of PREZISTA/ritonavir and artemether/lumefantrine can be used without dose adjustments. (bula de Darunavir, Interações medicamentosas)

  • Darunavir + cobicistateantirretroviralModerada

    Antimalarial: artemether/lumefantrine artemether: effect unknown lumefantrine: effect unknown Monitor for a potential decrease of antimalarial efficacy or potential QT prolongation. (bula de Darunavir + cobicistate, Interações medicamentosas)

  • Droperidolantagonista da dopaminaModerada

    Possible pharmacodynamic interactions can occur between droperidol and potentially arrhythmogenic agents such as class I or III antiarrhythmics, antihistamines that prolong the QT interval, antimalarials, calcium channel blockers, neuroleptics that prolong the QT interval, and antidepressants. (bula de Droperidol, Interações medicamentosas)

  • EfavirenzantirretroviralModerada

    Antimalarials: Artemether/lumefantrine Atovaquone/ proguanil ↓ artemether * ↓ dihydroartemisinin * ↓ lumefantrine * ↓ atovaquone ↓ proguanil Consider alternatives to artemether/ lumefantrine because of the risk of QT interval prolongation. (bula de Efavirenz, Interações medicamentosas)

  • Efavirenz + lamivudina + tenofovirantirretroviralModerada

    Antimalarials: Artemether/lumefantrine ↓ artemether ↓ dihydroartemisinin ↓ lumefantrine Consider alternatives to artemether/lumefantrine because of the risk of QT interval prolongation [see Warnings and Precautions (5.16) ] . (bula de Efavirenz + lamivudina + tenofovir, Interações medicamentosas)

  • EtravirinaantirretroviralModerada

    Antimalarial : artemether/lumefantrine ↔ etravirine ↓ artemether ↓ dihydroartemisinin ↓ lumefantrine Caution is warranted when co-administering Etravirine and artemether/lumefantrine as it is unknown whether the decrease in exposure of artemether or its active metabolite, dihydroartemisinin, could result in decreased antimalarial efficacy. (bula de Etravirina, Interações medicamentosas)

  • Hidroxicloroquinamedicamento que prolonga o intervalo QTModerada

    Co-administration of PLAQUENIL with other antimalarials known to lower the seizure threshold (e.g., mefloquine) may increase the risk of seizures. (bula de Hidroxicloroquina, Interações medicamentosas)

  • Lidocaína + epinefrinaanestésico localModerada

    Drugs Associated with Methemoglobinemia: Patients are at increased risk of developing methemoglobinemia when concurrently exposed to nitrates, nitrites, local anesthetics, antineoplastic agents, antibiotics, antimalarials, anticonvulsants, and other drugs. (bula de Lidocaína + epinefrina, Interações medicamentosas)

  • Lidocaína + prilocaínaanestésico localModerada

    …prilocaine, procaine, ropivacaine, tetracaine Antineoplastic agents cyclophosphamide, flutamide, hydroxyurea, isofamide, rasburicase Antibiotics dapsone, nitrofurantoin, para-aminosalicylic acid, sufonamides Antimalarials chloroquine, primaquine Anticonvulsants Phenobarbital, phenytoin, sodium valproate Other drugs acetaminophen, metoclopramide, quinine, sulfasalazine (bula de Lidocaína + prilocaína, Interações medicamentosas)

  • MefloquinaantimaláricoModerada

    Other Antimalarial Drugs Concomitant administration of mefloquine and other related antimalarial compounds (e.g., quinine, quinidine and chloroquine) may produce electrocardiographic abnormalities and increase the risk of convulsions (see WARNINGS ). (bula de Mefloquina, Interações medicamentosas)

  • Mepivacaínaanestésico localModerada

    …procaine, ropivacaine, tetracaine Antineoplastic agents cyclophosphamide, flutamide, hydroxyurea, ifosfamide, rasburicase Antibiotics dapsone, nitrofurantoin, para-aminosalicylic acid, sulfonamides Antimalarials chloroquine, primaquine Anticonvulsants phenobarbital, phenytoin, sodium valproate Other drugs acetaminophen, metoclopramide, quinine, sulfasalazine (bula de Mepivacaína, Interações medicamentosas)

  • Prilocaína + epinefrinaanestésico localModerada

    …ropivacaine, tetracaine Antineoplastic Agents cyclophosphamide, flutamide, hydroxyurea, ifosfamide, rasburicase Antibiotics dapsone, nitrofurantoin, para-aminosalicylic acid, sulfonamides Antimalarials chloroquine, primaquine Anticonvulsants phenobarbital, phenytoin, sodium valproate Other drugs acetaminophen, metoclopramide, quinine, sulfasalazine The administration… (bula de Prilocaína + epinefrina, Interações medicamentosas)

  • RifapentinaantibióticoModerada

    …quinidine, tocainide Antibiotics Chloramphenicol, clarithromycin, dapsone, doxycycline; Fluoroquinolones (such as ciprofloxacin) Oral Anticoagulants Warfarin Anticonvulsants Phenytoin Antimalarials Quinine Azole Antifungals Fluconazole, itraconazole, ketoconazole Antipsychotics Haloperidol Barbiturates Phenobarbital Benzodiazepines Diazepam Beta-Blockers Propranolol… (bula de Rifapentina, Interações medicamentosas)

  • Ropivacaínaanestésico localModerada

    …ropivacaine, tetracaine Antineoplastic agents cyclophosphamide, flutamide, hydroxyurea, ifosfamide, rasburicase Antibiotics dapsone, nitrofurantoin, para-aminosalicylic acid, sulfonamides Antimalarials chloroquine, primaquine Anticonvulsants Phenobarbital, phenytoin, sodium valproate Other drugs acetaminophen, metoclopramide, quinine, sulfasalazine NAROPIN should be… (bula de Ropivacaína, Interações medicamentosas)

Menções leves (3)

  • PirimetaminaantimaláricoLeve

    Drug Interactions: Pyrimethamine may be used with sulfonamides, quinine and other antimalarials, and with other antibiotics. (bula de Pirimetamina, Interações medicamentosas)

  • QuinidinaantiarrítmicoLeve

    Pediatric use In antimalarial trials, quinidine was as safe and effective in pediatric patients as in adults. (bula de Quinidina, Precauções)

  • QuininaantimaláricoLeve

    Other antimalarials (e.g., halofantrine, mefloquine). (bula de Quinina, Interações medicamentosas)

Verifique Tafenoquina com tudo o que você toma. Adicione sua lista completa; todos os pares são verificados de uma vez.

Abrir no verificador

Não é aconselhamento médico. A gravidade reflete a redação da bula, não as suas circunstâncias. Um alerta “grave” pode ser rotina sob supervisão, e um “leve” pode ser importante em doses altas. Pergunte a um farmacêutico.