Interacciones de Bexaroteno

Bexaroteno (Targretin), retinoide, tiene 58 interacciones documentadas en las etiquetas de la FDA y las hojas informativas que indexamos. Graves: 5; moderadas: 27; leves: 26; casos en los que una etiqueta indica que no hay ninguna interacción significativa: 0. Cada entrada de abajo cita la frase que la respalda. Esta página del medicamento es un punto de partida, no un veredicto sobre su situación.

Interacciones según la etiqueta

Interacciones graves (5)

  • AcitretinaretinoideGrave

    Acitretin is contraindicated in cases of hypersensitivity (e.g., angioedema, urticaria) to the preparation (acitretin or excipients) or to other retinoids . (etiqueta de Acitretina, Contraindicaciones)

  • GemfibrozilofibratoGrave

    Because of a potential drug-drug interaction, avoid gemfibrozil use with TARGRETIN [ see Drug Interactions (7) ]. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Minociclinaantibiótico del grupo de las tetraciclinasGrave

    Avoid concomitant use of isotretinoin and EMROSI because isotretinoin, a systemic retinoid, is also known to cause idiopathic intracranial hypertension. (etiqueta de Minociclina, Advertencias y precauciones)

  • Tetraciclinaantibiótico del grupo de las tetraciclinasGrave

    Concomitant use of isotretinoin and tetracycline should be avoided because isotretinoin, a systemic retinoid, is also known to cause pseudotumor cerebri. (etiqueta de Tetraciclina, Advertencias)

  • TretinoínaretinoideGrave

    Tretinoin capsules are contraindicated in patients with a known hypersensitivity to tretinoin capsules, any of its components, or other retinoids. (etiqueta de Tretinoína, Contraindicaciones)

Interacciones moderadas (27)

  • AlcoholAlcoholModerada

    Patients with CTCL who have risk factors for pancreatitis (e.g., prior pancreatitis, uncontrolled hyperlipidemia, excessive alcohol consumption, uncontrolled diabetes mellitus, biliary tract disease, and medications known to increase triglyceride levels or to be associated with pancreatic toxicity) may be at greater risk for pancreatitis associated with TARGRETIN… (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Drugs That Increase the Risk of Hypercalcemia Increase frequency of monitoring of calcium concentrations in patients taking concomitant Calcium Chloride Injection and other drugs that increase the risk of hypercalcemia (e.g., calcipotriene, estrogen, lithium, parathyroid hormone, teriparatide, thiazide diuretics, Vitamin A, and Vitamin D). (etiqueta de Cloruro de calcio, Interacciones medicamentosas)

  • Patients with elevated vitamin A levels may be at increased risk. (etiqueta de Elexacaftor, tezacaftor e ivacaftor, Advertencias y precauciones)

  • GlibenclamidasulfonilureaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Glibenclamida y metforminasulfonilureaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • GlimepiridasulfonilureaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • GlipizidasulfonilureaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Glipizida y metforminasulfonilureaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Insulina aspartainsulinaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Insulina degludecinsulinaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Insulina detemirinsulinaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Insulina glarginainsulinaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Insulina lisproinsulinaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Ivacaftorinhibidor de CYP3A4Moderada

    Patients with elevated vitamin A levels may be at increased risk. (etiqueta de Ivacaftor, Advertencias y precauciones)

  • Levotiroxinahormona tiroideaModerada

    Monitor and replace thyroid hormone if needed. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Levotiroxina y liotironinahormona tiroideaModerada

    Monitor and replace thyroid hormone if needed. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Liotironinahormona tiroideaModerada

    Monitor and replace thyroid hormone if needed. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Metimazolfármaco antitiroideoModerada

    Monitor and replace thyroid hormone if needed. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • MetotrexatoinmunosupresorModerada

    Monitor patients receiving XATMEP with other potential hepatotoxins (e.g., azathioprine, retinoids, and sulfasalazine) for possible signs of hepatotoxicity. (etiqueta de Metotrexato, Interacciones medicamentosas)

  • OrlistatModerada

    The effect of ORLISTAT on the absorption of supplemental vitamin D, vitamin A, and nutritionally-derived vitamin K is not known at this time [see Clinical Pharmacology (12.3) , and Warnings and Precautions (5.1) ] . (etiqueta de Orlistat, Interacciones medicamentosas)

  • PioglitazonatiazolidinedionaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Pioglitazona y glimepiridatiazolidinedionaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Pioglitazona y metforminatiazolidinedionaModerada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Propiltiouracilofármaco antitiroideoModerada

    Monitor and replace thyroid hormone if needed. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Teriparatidahormona tiroideaModerada

    Monitor and replace thyroid hormone if needed. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Tirzepatidaagonista del receptor de GLP-1Moderada

    Hypoglycemia Risk in Patients with Diabetes Mellitus In patients using insulin, agents enhancing insulin secretion (e.g., sulfonylureas), or insulin sensitizers (e.g., thiazolidinedione class), based on the mechanism of action, TARGRETIN could enhance the action of these agents, resulting in hypoglycemia. (etiqueta de Bexaroteno, Advertencias y precauciones)

Menciones leves (26)

  • Amlodipino y atorvastatinabloqueador de los canales de calcio dihidropiridínicoLeve

    Atorvastatin was used in 48% (73/152) of patients with CTCL. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • AtorvastatinaestatinaLeve

    Atorvastatin was used in 48% (73/152) of patients with CTCL. (etiqueta de Bexaroteno, Advertencias y precauciones)

  • Desogestrel y etinilestradiolanticonceptivo oralLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drospirenona y etinilestradiolanticonceptivo oralLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • EstradiolestrógenoLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Estradiol y dienogestanticonceptivo oralLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Fluconazolantifúngico azólicoLeve

    Vitamin A Based on a case report in one patient receiving combination therapy with all-trans-retinoid acid (an acid form of vitamin A) and fluconazole, central nervous system (CNS) related undesirable effects have developed in the form of pseudotumor cerebri, which disappeared after discontinuation of fluconazole treatment. (etiqueta de Fluconazol, Interacciones medicamentosas)

  • FulvestrantestrógenoLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drugs that may cause hypercalcemia: Vitamin D, vitamin A, thiazide diuretics, estrogen, calcipotriene and teriparatide administration may cause hypercalcemia. (etiqueta de Gluconato de calcio, Interacciones medicamentosas)

  • LevonorgestrelprogestágenoLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Levonorgestrel y etinilestradiolanticonceptivo oralLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • MedroxiprogesteronaprogestágenoLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • MegestrolprogestágenoLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Mifepristonainhibidor de CYP3A4Leve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • NoretisteronaprogestágenoLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Noretisterona y etinilestradiolanticonceptivo oralLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Norgestimato y etinilestradiolanticonceptivo oralLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • Norgestrel y etinilestradiolanticonceptivo oralLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

  • ProgesteronaprogestágenoLeve

    Drug products which may be affected include oral or other systemic hormonal contraceptives. (etiqueta de Bexaroteno, Interacciones medicamentosas)

Compruebe Bexaroteno frente a todo lo que toma. Añada su lista completa; todos los pares se comprueban a la vez.

Abrir en el verificador

No es un consejo médico. La gravedad refleja la redacción de la etiqueta, no sus circunstancias. Una señal «grave» puede ser algo habitual bajo supervisión y una «leve» puede ser importante a dosis altas. Consulte a un farmacéutico.