Interações de Danazol

Danazol, androgênio, tem 80 interações documentadas nas bulas da FDA e nas fichas informativas que indexamos (graves: 6; moderadas: 73; leves: 1; casos em que uma bula relata não haver interação significativa: 0). Cada item abaixo cita a frase em que se baseia. Esta página de medicamento é um ponto de partida, não um veredito para a sua situação.

Interações segundo a bula

Interações graves (6)

  • DoravirinaantirretroviralGrave

    These drugs include, but are not limited to, the following: the anticonvulsants carbamazepine, oxcarbazepine, phenobarbital, phenytoin the androgen receptor inhibitor enzalutamide the antimycobacterials rifampin, rifapentine the cytotoxic agent mitotane St. (bula de Doravirina, Contraindicações)

  • Concomitant use of cyclosporine, danazol, or danazol [see Drug Interactions (7.1) ] . (bula de Ezetimiba + sinvastatina, Contraindicações)

  • Finasteridainibidor da 5-alfa-redutaseGrave

    Because of the ability of Type II 5α-reductase inhibitors to inhibit the conversion of testosterone to 5α-dihydrotestosterone (DHT), finasteride may cause abnormalities of the external genitalia of a male fetus of a pregnant female who receives finasteride. (bula de Finasterida, Contraindicações)

  • CONTRAINDICATIONS: Precocious puberty, prostatic carcinoma or other androgen-dependent neoplasm, prior allergic reaction to HCG. (bula de Gonadotrofina coriônica, Contraindicações)

  • LovastatinaestatinaGrave

    …Voriconazole Erythromycin Clarithromycin Telithromycin HIV protease inhibitors Boceprevir Telaprevir Nefazodone Cobicistat-containing products Gemfibrozil Avoid with lovastatin Cyclosporine Danazol Do not exceed 20 mg lovastatin daily Diltiazem Dronedarone Verapamil Amiodarone Do not exceed 40 mg lovastatin daily Grapefruit juice Avoid grapefruit juice Immune-Mediated… (bula de Lovastatina, Advertências)

  • SinvastatinaestatinaGrave

    Concomitant use of cyclosporine, danazol or gemfibrozil [see Drug Interactions (7.1) ] . (bula de Sinvastatina, Contraindicações)

Interações moderadas (73)

  • AcarboseantidiabéticoModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • PRECAUTIONS General Induction of androgen secretion by hCG may cause fluid retention. (bula de Alfacoriogonadotropina, Precauções)

  • Alogliptinainibidor da DPP-4Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Alogliptina + metforminainibidor da DPP-4Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Anlodipino + atorvastatinabloqueador dos canais de cálcio di-hidropiridínicoModerada

    The risk of myopathy and rhabdomyolysis is increased by concomitant administration of danazol with statins such as simvastatin, atorvastatin and lovastatin. (bula de Danazol, Interações medicamentosas)

  • AtorvastatinaestatinaModerada

    The risk of myopathy and rhabdomyolysis is increased by concomitant administration of danazol with statins such as simvastatin, atorvastatin and lovastatin. (bula de Danazol, Interações medicamentosas)

  • Bexagliflozinainibidor do SGLT2Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Calcipotriolanálogo da vitamina DModerada

    Danazol can increase the calcemic response to synthetic vitamin D analogs in primary hypoparathyroidism. (bula de Danazol, Interações medicamentosas)

  • Calcitriolanálogo da vitamina DModerada

    Danazol can increase the calcemic response to synthetic vitamin D analogs in primary hypoparathyroidism. (bula de Danazol, Interações medicamentosas)

  • Canagliflozinainibidor do SGLT2Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • CarbamazepinaanticonvulsivanteModerada

    Therapy with danazol may cause an increase in carbamazepine levels in patients taking both drugs. (bula de Danazol, Interações medicamentosas)

  • CiclosporinaimunossupressorModerada

    …methylprednisolone Allopurinol nicardipine itraconazole clarithromycin Amiodarone verapamil ketoconazole erythromycin Bromocriptine voriconazole quinupristin/ dalfopristin colchicine danazol imatinib metoclopramide nefazodone oral contraceptives HIV Protease Inhibitors The HIV protease inhibitors (e.g., indinavir, nelfinavir, ritonavir, and saquinavir) are known… (bula de Ciclosporina, Interações medicamentosas)

  • Dapagliflozinainibidor do SGLT2Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Dapagliflozina + metforminainibidor do SGLT2Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Doxercalciferolanálogo da vitamina DModerada

    Danazol can increase the calcemic response to synthetic vitamin D analogs in primary hypoparathyroidism. (bula de Danazol, Interações medicamentosas)

  • Dulaglutidaagonista do receptor de GLP-1Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Empagliflozinainibidor do SGLT2Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Empagliflozina + metforminainibidor do SGLT2Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Espironolactona + hidroclorotiazidaantagonista da aldosteronaModerada

    Abiraterone: Spironolactone binds to the androgen receptor and may increase prostate‑specific antigen (PSA) levels in abiraterone-treated prostate cancer patients. (bula de Espironolactona + hidroclorotiazida, Interações medicamentosas)

  • Estradiol + noretisteronaestrogênioModerada

    Free hormone concentrations, such as testosterone and estradiol, may be decreased. (bula de Estradiol + noretisterona, Advertências e precauções)

  • Estrogênios conjugadosestrogênioModerada

    Free hormone concentrations, such as testosterone and estradiol, may be decreased. (bula de Estrogênios conjugados, Precauções)

  • Free hormone concentrations, such as testosterone and estradiol, may be decreased. (bula de Estrogênios conjugados + bazedoxifeno, Advertências e precauções)

  • Exenatidaagonista do receptor de GLP-1Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • FludrocortisonacorticosteroideModerada

    Anabolic steroids (particularly C-17 alkylated androgens such as oxymetholone, methandrostenolone, norethandrolone, and similar compounds)—enhanced tendency toward edema. (bula de Fludrocortisona, Interações medicamentosas)

  • FluvastatinaestatinaModerada

    The risk of myopathy and rhabdomyolysis is increased by concomitant administration of danazol with statins such as simvastatin, atorvastatin and lovastatin. (bula de Danazol, Interações medicamentosas)

  • FolitropinaModerada

    For Men : Clinical monitoring for spermatogenesis utilizes the following indirect or direct measures: Serum testosterone level Semen analysis 5.11 FOLLISTIM Pen The FOLLISTIM Pen is intended only for use with FOLLISTIM AQ Cartridge. (bula de Folitropina, Advertências e precauções)

  • GlibenclamidasulfonilureiaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Glibenclamida + metforminasulfonilureiaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • GlimepiridasulfonilureiaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • GlipizidasulfonilureiaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Glipizida + metforminasulfonilureiaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • GosserrelinaModerada

    Effect on QT/QTc Interval: Androgen deprivation therapy may prolong the QT interval. (bula de Gosserrelina, Advertências e precauções)

  • Insulina asparteinsulinaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Insulina degludecainsulinaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Insulina detemirinsulinaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Insulina glarginainsulinaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Insulina lisproinsulinaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Tumor Flare: Increased serum testosterone (~ 50% above baseline) may occur when initiating treatment with LUPRON DEPOT. (bula de Leuprorrelina, Advertências e precauções)

  • Levotiroxinahormônio tireoidianoModerada

    Other metabolic events include a reduction in thyroid binding globulin and T4 with increased uptake of T3, but without disturbance of thyroid stimulating hormone or of free thyroxin index. (bula de Danazol, Precauções)

  • Levotiroxina + liotironinahormônio tireoidianoModerada

    Other metabolic events include a reduction in thyroid binding globulin and T4 with increased uptake of T3, but without disturbance of thyroid stimulating hormone or of free thyroxin index. (bula de Danazol, Precauções)

  • Linagliptinainibidor da DPP-4Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Linagliptina + metforminainibidor da DPP-4Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Liotironinahormônio tireoidianoModerada

    Other metabolic events include a reduction in thyroid binding globulin and T4 with increased uptake of T3, but without disturbance of thyroid stimulating hormone or of free thyroxin index. (bula de Danazol, Precauções)

  • Liraglutidaagonista do receptor de GLP-1Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • MedroxiprogesteronaprogestinaModerada

    The following laboratory tests may be affected by progestins including MPA Injectable Suspension, USP: (a) Plasma and urinary steroid levels are decreased (e.g., progesterone, estradiol, pregnanediol, testosterone, cortisol). (bula de Medroxiprogesterona, Interações medicamentosas)

  • MetforminabiguanidaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • MiglitolantidiabéticoModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • NateglinidameglitinidaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Paricalcitolanálogo da vitamina DModerada

    Danazol can increase the calcemic response to synthetic vitamin D analogs in primary hypoparathyroidism. (bula de Danazol, Interações medicamentosas)

  • PioglitazonatiazolidinedionaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Pioglitazona + glimepiridatiazolidinedionaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Pioglitazona + metforminatiazolidinedionaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • PitavastatinaestatinaModerada

    The risk of myopathy and rhabdomyolysis is increased by concomitant administration of danazol with statins such as simvastatin, atorvastatin and lovastatin. (bula de Danazol, Interações medicamentosas)

  • PravastatinaestatinaModerada

    The risk of myopathy and rhabdomyolysis is increased by concomitant administration of danazol with statins such as simvastatin, atorvastatin and lovastatin. (bula de Danazol, Interações medicamentosas)

  • Propiltiouracilamedicamento antitireoidianoModerada

    Other metabolic events include a reduction in thyroid binding globulin and T4 with increased uptake of T3, but without disturbance of thyroid stimulating hormone or of free thyroxin index. (bula de Danazol, Precauções)

  • Ramelteonasedativo-hipnóticoModerada

    Reproductive effects: Include decreased testosterone and increased prolactin levels. (bula de Ramelteona, Advertências e precauções)

  • RepaglinidameglitinidaModerada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • RosuvastatinaestatinaModerada

    The risk of myopathy and rhabdomyolysis is increased by concomitant administration of danazol with statins such as simvastatin, atorvastatin and lovastatin. (bula de Danazol, Interações medicamentosas)

  • Saxagliptinainibidor da DPP-4Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Saxagliptina + metforminainibidor da DPP-4Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Semaglutidaagonista do receptor de GLP-1Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • SirolimoimunossupressorModerada

    • Drugs that could increase sirolimus blood concentrations: Bromocriptine, cimetidine, cisapride, clotrimazole, danazol, diltiazem, fluconazole, letermovir, protease inhibitors (e.g., HIV and hepatitis C that include drugs such as ritonavir, indinavir, boceprevir, and telaprevir), metoclopramide, nicardipine, troleandomycin, verapamil • Drugs and other agents… (bula de Sirolimo, Interações medicamentosas)

  • Sitagliptinainibidor da DPP-4Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Sitagliptina + metforminainibidor da DPP-4Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • TacrolimoimunossupressorModerada

    Danazol may raise the plasma levels of cyclosporin and tacrolimus, leading to an increase of the renal toxicity of these drugs. (bula de Danazol, Interações medicamentosas)

  • Tamoxifenomodulador seletivo do receptor de estrogênioModerada

    Hypercalcemia in Patients with Metastatic Breast Cancer As with other additive hormonal therapy (estrogens and androgens), hypercalcemia has been reported in some breast cancer patients with bone metastases within a few weeks of starting treatment with tamoxifen. (bula de Tamoxifeno, Advertências e precauções)

  • Teriparatidahormônio tireoidianoModerada

    Other metabolic events include a reduction in thyroid binding globulin and T4 with increased uptake of T3, but without disturbance of thyroid stimulating hormone or of free thyroxin index. (bula de Danazol, Precauções)

  • Tiamazol (metimazol)medicamento antitireoidianoModerada

    Other metabolic events include a reduction in thyroid binding globulin and T4 with increased uptake of T3, but without disturbance of thyroid stimulating hormone or of free thyroxin index. (bula de Danazol, Precauções)

  • Tirzepatidaagonista do receptor de GLP-1Moderada

    Caution should be exercised when used with antidiabetic drugs. (bula de Danazol, Interações medicamentosas)

  • Tumor Flare: Transient increase in serum testosterone levels can occur within the first few weeks of treatment. (bula de Triptorrelina, Advertências e precauções)

  • VarfarinaanticoagulanteModerada

    Drug Interactions: Prolongation of prothrombin time occurs in patients stabilized on warfarin. (bula de Danazol, Interações medicamentosas)

  • Vitamina DVitaminas e mineraisModerada

    Danazol can increase the calcemic response to synthetic vitamin D analogs in primary hypoparathyroidism. (bula de Danazol, Interações medicamentosas)

Menções leves (1)

  • TestosteronaandrogênioLeve

    Laboratory Tests: Danazol treatment may interfere with laboratory determinations of testosterone, androstenedione and dehydroepiandrosterone. (bula de Danazol, Precauções)

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