Interações de Tigeciclina

Tigeciclina (Tygacil), antibiótico da classe das tetraciclinas, tem 61 interações documentadas nas bulas da FDA e nas fichas informativas que indexamos (graves: 8; moderadas: 19; leves: 31; casos em que uma bula relata não haver interação significativa: 3). Cada item abaixo cita a frase em que se baseia. Esta página de medicamento é um ponto de partida, não um veredito para a sua situação.

Interações segundo a bula

Interações graves (8)

  • AcitretinaretinoideGrave

    Since both acitretin and tetracyclines can cause increased intracranial pressure, their combined use is contraindicated (see WARNINGS: Pseudotumor Cerebri ). (bula de Acitretina, Contraindicações)

  • Benzilpenicilina (penicilina G)antibiótico da classe das penicilinasGrave

    Drug Interactions Bacteriostatic antibacterials ( i.e. , chloramphenicol, erythromycins, sulfonamides or tetracyclines) may antagonize the bactericidal effect of penicillin, and concurrent use of these drugs should be avoided. (bula de Benzilpenicilina (penicilina G), Interações medicamentosas)

  • CiclosporinaimunossupressorGrave

    Therefore, serum concentrations of the calcineurin inhibitor should be monitored during treatment with TYGACIL to avoid drug toxicity. (bula de Tigeciclina, Interações medicamentosas)

  • IsotretinoínaretinoideGrave

    Intracranial Hypertension ( Pseudotumor Cerebri ): Avoid concomitant use with tetracyclines ( 5.5 ) (bula de Isotretinoína, Advertências e precauções)

  • Pimecrolimoinibidor da calcineurinaGrave

    Therefore, serum concentrations of the calcineurin inhibitor should be monitored during treatment with TYGACIL to avoid drug toxicity. (bula de Tigeciclina, Interações medicamentosas)

  • Avoid use in patients with known hypersensitivity to tetracyclines. (bula de Tigeciclina, Advertências e precauções)

  • TacrolimoimunossupressorGrave

    Therefore, serum concentrations of the calcineurin inhibitor should be monitored during treatment with TYGACIL to avoid drug toxicity. (bula de Tigeciclina, Interações medicamentosas)

  • Tetraciclinaantibiótico da classe das tetraciclinasGrave

    Avoid use in patients with known hypersensitivity to tetracyclines. (bula de Tigeciclina, Advertências e precauções)

Interações moderadas (19)

  • Acetato de cálcioquelante de fosfatoModerada

    Calcium acetate capsules may decrease the bioavailability of tetracyclines or fluoroquinolones via this mechanism. (bula de Acetato de cálcio, Interações medicamentosas)

  • AtovaquonaantimaláricoModerada

    • Concomitant administration of tetracycline reduces atovaquone concentrations; use caution when coadministering. (bula de Atovaquona, Interações medicamentosas)

  • Atovaquona + proguanilantimaláricoModerada

    • Tetracycline may reduce atovaquone concentrations; parasitemia should be closely monitored. (bula de Atovaquona + proguanil, Interações medicamentosas)

  • CálcioVitaminas e mineraisModerada

    O cálcio se liga a esses medicamentos no intestino e pode reduzir drasticamente a quantidade absorvida; separe as doses. (NIH Office of Dietary Supplements, Calcium)

  • Colestipolsequestrante de ácidos biliaresModerada

    The absorption of tetracycline, furosemide, penicillin G, hydrochlorothiazide, and gemfibrozil was significantly decreased when given simultaneously with colestipol hydrochloride; these drugs were not tested to determine the effect of administration one hour before colestipol hydrochloride. (bula de Colestipol, Interações medicamentosas)

  • Colestiraminasequestrante de ácidos biliaresModerada

    Drug Interactions Cholestyramine for Oral Suspension USP may delay or reduce the absorption of concomitant oral medication such as phenylbutazone, warfarin, thiazide diuretics (acidic), or propranolol (basic), as well as tetracycline, penicillin G, phenobarbital, thyroid and thyroxine preparations, estrogens and progestins, and digitalis. (bula de Colestiramina, Interações medicamentosas)

  • FerroVitaminas e mineraisModerada

    O ferro se liga a esses medicamentos no intestino e reduz a sua absorção; separe as doses. (NIH Office of Dietary Supplements, Iron)

  • GlimepiridasulfonilureiaModerada

    …antagonists, fibrates, propoxyphene, pentoxifylline, somatostatin analogs, anabolic steroids and androgens, cyclophosphamide, phenyramidol, guanethidine, fluconazole, sulfinpyrazone, tetracyclines, clarithromycin, disopyramide, quinolones, and those drugs that are highly protein-bound, such as fluoxetine, nonsteroidal anti-inflammatory drugs, salicylates, sulfonamides,… (bula de Glimepirida, Interações medicamentosas)

  • Lantânioquelante de fosfatoModerada

    Examples of relevant classes of compounds where antacids have been demonstrated to reduce bioavailability include antibiotics (such as quinolones, ampicillin, and tetracyclines), thyroid hormones, ACE inhibitors, statin lipid regulators, and anti-malarials. (bula de Lantânio, Interações medicamentosas)

  • LomitapidaModerada

    Caution should be exercised when JUXTAPID is used with other medications known to have potential for hepatotoxicity, such as isotretinoin, amiodarone, acetaminophen (>4 g/day for ≥3 days/week), methotrexate, tetracyclines, and tamoxifen. (bula de Lomitapida, Advertências e precauções)

  • MagnésioVitaminas e mineraisModerada

    Suplementos e antiácidos que contêm magnésio reduzem a absorção desses medicamentos; separe as doses em pelo menos duas horas. (NIH Office of Dietary Supplements, Magnesium)

  • Pioglitazona + glimepiridatiazolidinedionaModerada

    …antagonists, fibrates, propoxyphene, pentoxifylline, somatostatin analogs, anabolic steroids and androgens, cyclophosphamide, phenyramidol, guanethidine, fluconazole, sulfinpyrazone, tetracyclines, clarithromycin, disopyramide, quinolones, and those drugs that are highly protein-bound, such as fluoxetine, nonsteroidal anti-inflammatory drugs, salicylates, sulfonamides,… (bula de Pioglitazona + glimepirida, Interações medicamentosas)

  • Quinaprilinibidor da ECAModerada

    Tetracycline and other drugs that interact with magnesium Simultaneous administration of tetracycline with quinapril hydrochloride reduced the absorption of tetracycline by approximately 28% to 37%, possibly due to the high magnesium content in quinapril tablets. (bula de Quinapril, Interações medicamentosas)

  • QuininaantimaláricoModerada

    Although tetracycline may be concomitantly administered with quinine sulfate, patients should be monitored closely for adverse reactions associated with quinine sulfate. (bula de Quinina, Interações medicamentosas)

  • Rocurôniobloqueador neuromuscularModerada

    Antibiotics Drugs which may enhance the neuromuscular blocking action of nondepolarizing agents such as Rocuronium Bromide Injection include certain antibiotics (e.g., aminoglycosides; vancomycin; tetracyclines; bacitracin; polymyxins; colistin; and sodium colistimethate). (bula de Rocurônio, Interações medicamentosas)

  • SucralfatoModerada

    Drug Interactions Some studies have shown that simultaneous sucralfate administration in healthy volunteers reduced the extent of absorption (bioavailability) of single doses of the following: cimetidine, digoxin, fluoroquinolone antibiotics, ketoconazole, l-thyroxine, phenytoin, quinidine, ranitidine, tetracycline, and theophylline. (bula de Sucralfato, Interações medicamentosas)

  • TretinoínaretinoideModerada

    The concomitant use of other products (e.g., tetracyclines) that can cause intracranial hypertension may increase the risk. (bula de Tretinoína, Advertências e precauções)

  • VarfarinaanticoagulanteModerada

    • Warfarin : Suitable anticoagulation test should be monitored if TYGACIL is administered to patients receiving warfarin. (bula de Tigeciclina, Interações medicamentosas)

  • ZincoVitaminas e mineraisModerada

    O zinco reduz a absorção dos antibióticos das classes das quinolonas e das tetraciclinas; tome o antibiótico pelo menos duas horas antes ou quatro a seis horas depois do zinco. (NIH Office of Dietary Supplements, Zinc)

Menções leves (31)

  • Amoxicilinaantibiótico da classe das penicilinasLeve

    Other Antibacterials Chloramphenicol, macrolides, sulfonamides, and tetracyclines may interfere with the bactericidal effects of penicillin. (bula de Amoxicilina, Interações medicamentosas)

  • Ampicilinaantibiótico da classe das penicilinasLeve

    Bacteriostatic Antibiotics : Chloramphenicol, erythromycins, sulfonamides, or tetracyclines may interfere with the bactericidal effect of penicillins. (bula de Ampicilina, Interações medicamentosas)

  • Demeclociclinaantibiótico da classe das tetraciclinasLeve

    WARNINGS DEMECLOCYCLINE HYDROCHLORIDE, LIKE OTHER TETRACYCLINE-CLASS ANTIBIOTICS, CAN CAUSE FETAL HARM WHEN ADMINISTERED TO A PREGNANT WOMAN. (bula de Demeclociclina, Advertências)

  • Desogestrel + etinilestradiolanticoncepcional oralLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Dicloxacilinaantibiótico da classe das penicilinasLeve

    Drug Interactions Tetracycline, a bacteriostatic antibiotic, may antagonize the bactericidal effect of penicillin and concurrent use of these drugs should be avoided. (bula de Dicloxacilina, Interações medicamentosas)

  • Drospirenona + etinilestradiolanticoncepcional oralLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • EstradiolestrogênioLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Estradiol + dienogesteanticoncepcional oralLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • FulvestrantoestrogênioLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • HeparinaanticoagulanteLeve

    Other Interactions Digitalis, tetracyclines, nicotine, or antihistamines, or intravenous nitroglycerin may partially counteract the anticoagulant action of heparin sodium. (bula de Heparina, Interações medicamentosas)

  • Imipeném + cilastatinaantibióticoLeve

    In cIAI studies (n=1642), 6 patients treated with TYGACIL and 2 patients treated with imipenem/cilastatin presented with intestinal perforations and developed sepsis/septic shock. (bula de Tigeciclina, Advertências e precauções)

  • LevonorgestrelprogestinaLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Levonorgestrel + etinilestradiolanticoncepcional oralLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • MedroxiprogesteronaprogestinaLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • MegestrolprogestinaLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Mifepristonainibidor da CYP3A4Leve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Nafcilinaantibiótico da classe das penicilinasLeve

    Drug Interactions Tetracycline, a bacteriostatic antibiotic, may antagonize the bactericidal effect of penicillin, and concurrent use of these drugs should be avoided. (bula de Nafcilina, Interações medicamentosas)

  • Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • NoretisteronaprogestinaLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Noretisterona + etinilestradiolanticoncepcional oralLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Norgestimato + etinilestradiolanticoncepcional oralLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Norgestrel + etinilestradiolanticoncepcional oralLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Oxacilinaantibiótico da classe das penicilinasLeve

    Drug Interactions Tetracycline, a bacteriostatic antibiotic, may antagonize the bactericidal effect of penicillin and concurrent use of these drugs should be avoided. (bula de Oxacilina, Interações medicamentosas)

  • ProgesteronaprogestinaLeve

    Oral Contraceptives Concurrent use of antibacterial drugs with oral contraceptives may render oral contraceptives less effective. (bula de Tigeciclina, Interações medicamentosas)

  • Vecurôniobloqueador neuromuscularLeve

    The following antibiotics have been associated with various degrees of paralysis: aminoglycosides (such as neomycin, streptomycin, kanamycin, gentamicin, and dihydrostreptomycin); tetracyclines; bacitracin; polymyxin B; colistin; and sodium colistimethate. (bula de Vecurônio, Precauções)

Nenhuma interação significativa relatada (3)

  • AminofilinametilxantinaSem interação

    …omeprazole prednisone, prednisolone ranitidine rifabutin roxithromycin sorbitol (purgative doses do not inhibit theophylline absorption) sucralfate terbutaline, systemic terfenadine tetracycline tocainide The Effect of Other Drugs on Theophylline Serum Concentration Measurements: Most serum theophylline assays in clinical use are immunoassays which are specific… (bula de Aminofilina, Interações medicamentosas)

  • Cisatracúriobloqueador neuromuscularSem interação

    …additional doses of Cisatracurium Besylate Injection, and to determine whether adjustments need to be made to the dose with subsequent administration. † Examples: aminoglycosides, tetracyclines, bacitracin, polymyxins, lincomycin, clindamycin, colistin, sodium colistimethate Drug or Drug Class Clinical Implications * Succinylcholine The use of succinylcholine… (bula de Cisatracúrio, Interações medicamentosas)

  • TeofilinametilxantinaSem interação

    …ranitidine famotidine rifabutin felodipine roxithromycin finasteride Sorbitol (purgative doses do not inhibit hydrocortisone theophylline absorption) isoflurane sucralfate isoniazid terbutaline, systemic isradipine terfenadine influenza vaccine tetracycline ketoconazole tocainide lomefloxacin * Refer to PRECAUTIONS , Drug Interactions for information regarding table. (bula de Teofilina, Interações medicamentosas)

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Não é aconselhamento médico. A gravidade reflete a redação da bula, não as suas circunstâncias. Um alerta “grave” pode ser rotina sob supervisão, e um “leve” pode ser importante em doses altas. Pergunte a um farmacêutico.